Wednesday, November 18, 2009

5-Fluorouracil

Pyrimidine antimetabolite used for colon, rectum, gastric, pancreatic and breast cancer.
- Inhibits thymidylate synthase which prevents DNA and RNA synthesis.  Enhanced by addition of leucovorin.

Side-effects:
- mucositis, diarrhea from epithelial cell turnover.
- hand-foot syndrome
- myelosuppression less with continuous infusions

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